SCHEMBL6990547

SCHEMBL6990547

NS(=O)(=O)c1ccc(C2=C(c3cccc(F)c3)C(=O)OC23CCC3)cc1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.56
PTGS1 P23219 9/20 0.56
CA12 O43570 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
CA1 P00915 1/20 0.40
CHRNA7 P36544 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990787 0.98 PTGS2 (0.56) PTGS2PTGS1CA12CA2CA9
SCHEMBL6990070 0.89 PTGS2 (0.71) PTGS2PTGS1
SCHEMBL6990691 0.88 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL6987745 0.87 PTGS2 (0.53) PTGS2PTGS1CA2CA1
SCHEMBL6992321 0.86 PTGS2 (0.71) PTGS2PTGS1
SCHEMBL6990955 0.86 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL6989032 0.86 PTGS2 (0.54) PTGS2PTGS1CA12CA2CA9
SCHEMBL6994862 0.85 PTGS2 (0.53) PTGS2PTGS1CA2CA1
SCHEMBL6995595 0.85 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL6994660 0.84 PTGS2 (0.74) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799218-B1 DIARYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2003-02-19 EP claimed
US-6222048-B1 AS ANTIINFLAMMATORY, ANTIPYRETIC AND ANALGESIC AGENTS; INHIBITS HORMONE INDUCED UTERINE CONTRACTION; ANTICANCER PROPERTIES; SIDE EFFECT REDUCTION MERCK FROSST CANADA & CO. (CA) 2001-04-24 US claimed
EP-0799218-B1 DIARYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2003-02-19 EP disclosed
US-6222048-B1 AS ANTIINFLAMMATORY, ANTIPYRETIC AND ANALGESIC AGENTS; INHIBITS HORMONE INDUCED UTERINE CONTRACTION; ANTICANCER PROPERTIES; SIDE EFFECT REDUCTION MERCK FROSST CANADA & CO. (CA) 2001-04-24 US disclosed