SCHEMBL6990584

SCHEMBL6990584

O=C(NCc1ccccc1)c1cc2ccccc2c(Cl)n1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.56
LCK P06239 1/20 0.56
MMP13 P45452 1/20 0.56
NPC1 O15118 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C19 P33261 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
ALDH1A1 P00352 4/20 0.52
HPGD P15428 3/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
POLB P06746 1/20 0.50
RAB9A P51151 1/20 0.49
GLA P06280 1/20 0.49
TP53 P04637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10982335 0.82 CNR1 (0.56) EGFRLCKMMP13MEN1KMT2A
SCHEMBL30023908 0.78 KDM4E (0.50) CYP1A2CYP2C19MEN1KMT2AALDH1A1
SCHEMBL1990776 0.78 KDM4E (0.50) CYP1A2CYP2C19MEN1KMT2AALDH1A1
SCHEMBL20606513 0.75 EGFR (0.59) EGFRLCKMMP13CYP1A2CYP2D6
SCHEMBL11640078 0.75 TSHR (0.60) EGFRMMP13NPC1CYP1A2CYP2C19
SCHEMBL21753196 0.75 HPGD (0.79) EGFRMMP13CYP1A2CYP2D6CYP2C19
SCHEMBL12447827 0.73 NPC1 (0.49) NPC1MEN1KMT2APOLBRAB9A
SCHEMBL3281702 0.73 KDM4E (0.50) LCKNPC1CYP1A2CYP2C19MEN1
SCHEMBL8975296 0.73 BCHE (0.72) MMP13NPC1MEN1KMT2AALDH1A1
SCHEMBL6491776 0.72 MMP13 (0.61) EGFRMMP13CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023268-B1 ISOQUINOLINES AS UROKINASE INHIBITORS PFIZER LTD (GB) 2003-05-21 EP disclosed