SCHEMBL6990754

SCHEMBL6990754

Cc1cccc(Cl)c1CNc1ccc(-c2c(C#N)[nH]c3ccccc23)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 4/20 0.41
PDE1C Q14123 1/20 0.41
ABL1 P00519 1/20 0.37
SRC P12931 1/20 0.37
CYP3A4 P08684 1/20 0.37
CD38 P28907 1/20 0.37
EIF2AK1 Q9BQI3 2/20 0.35
KMT2A Q03164 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PLA2G1B P04054 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ATG4B Q9Y4P1 1/20 0.34
ADRA2B P18089 1/20 0.34
GCGR P47871 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989051 0.87 RXFP1 (0.46) PDE9APDE1CCD38KMT2AGAA
SCHEMBL4926760 0.72 MAPT (0.47) ABL1SRCCYP3A4CD38EIF2AK1
SCHEMBL6986759 0.71 PDE9A (0.35) PDE9APDE1CKMT2ANPC1RAB9A
SCHEMBL11552943 0.70 PDE9A (0.61) PDE9APDE1CCYP3A4KMT2AGAA
SCHEMBL6989632 0.66 GAA (0.40) PDE9APDE1CABL1SRCKMT2A
SCHEMBL6987924 0.66 PDE9A (0.37) PDE9APDE1CABL1CYP3A4
SCHEMBL6988191 0.65 MAPT (0.41) ABL1SRCCYP3A4CD38EIF2AK1
SCHEMBL10061644 0.62 P2RX7 (0.44) CYP3A4CD38EIF2AK1KMT2AKDM4E
SCHEMBL4943568 0.62 MAPT (0.56) KMT2ARAB9AGAAKDM4EALDH1A1
SCHEMBL3680016 0.61 AHR (0.55) PDE9APDE1CSRCCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303508-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2003-04-23 EP claimed
WO-2002006273-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-01-24 WO claimed