SCHEMBL6990854

SCHEMBL6990854

O=C1c2c(ccn2Cc2ccccc2)/C(=N\O)CCN1CCCN1CCN(c2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.46
DRD3 P35462 8/20 0.44
DRD2 P14416 5/20 0.44
DRD5 P21918 1/20 0.44
HTR7 P34969 2/20 0.44
DRD4 P21917 2/20 0.43
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
SIGMAR1 Q99720 2/20 0.42
DRD1 P21728 2/20 0.42
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
HTR2A P28223 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990858 1.00 HTR1A (0.46) HTR1ADRD3DRD2DRD5HTR7
SCHEMBL6993434 0.91 HTR1A (0.46) HTR1ADRD3DRD2DRD5HTR7
SCHEMBL6993431 0.91 HTR1A (0.46) HTR1ADRD3DRD2DRD5HTR7
SCHEMBL6993124 0.88 HTR1A (0.49) HTR1ADRD3DRD2DRD5HTR7
SCHEMBL6992608 0.87 HTR1A (0.48) HTR1ADRD3DRD2DRD5HTR7
SCHEMBL6992602 0.87 HTR1A (0.48) HTR1ADRD3DRD2DRD5HTR7
SCHEMBL6989075 0.85 HTR1A (0.49) HTR1ADRD3DRD2DRD5HTR7
SCHEMBL6989077 0.85 HTR1A (0.49) HTR1ADRD3DRD2DRD5HTR7
SCHEMBL7140268 0.82 HTR1A (0.48) HTR1ADRD3DRD2DRD5HTR7
SCHEMBL7140269 0.82 HTR1A (0.48) HTR1ADRD3DRD2DRD5HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557526-B1 PYRROLOAZEPINE COMPOUND SUNTORY LTD (JP) 2003-04-02 EP disclosed
US-5399557-A Cardiovascular disorders SUNTORY LIMITED (JP) 1995-03-21 US disclosed
EP-0557526-A1 PYRROLOAZEPINE COMPOUND SUNTORY LIMITED (JP) 1993-09-01 EP disclosed