SCHEMBL6990967

SCHEMBL6990967

CN(C)C(=O)c1ccc(Nc2ncc3ncnc(Nc4ccc(F)c(Cl)c4)c3n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.56
ERBB2 P04626 7/20 0.56
HPGD P15428 1/20 0.56
HTT P42858 1/20 0.56
AURKA O14965 1/20 0.55
CSNK2A1 P68400 3/20 0.50
USP2 O75604 1/20 0.49
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
MAPT P10636 1/20 0.49
ERBB4 Q15303 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
BRAF P15056 1/20 0.47
GRM1 Q13255 1/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990337 0.89 EGFR (0.56) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8317835 0.86 EGFR (0.56) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8487596 0.83 EGFR (0.59) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL6993963 0.83 EGFR (0.56) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8484377 0.82 EGFR (0.64) EGFRERBB2HPGDHTTAURKA
SCHEMBL6992430 0.82 EGFR (0.62) EGFRERBB2HPGDHTTMAPT
SCHEMBL6992426 0.81 EGFR (0.53) EGFRERBB2HPGDHTTAURKA
SCHEMBL8488002 0.81 LRRK2 (0.57) EGFRERBB2HPGDHTTMAPT
SCHEMBL8314458 0.80 EGFR (0.53) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8318976 0.80 EGFR (0.54) EGFRERBB2HPGDHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888351-B1 PYRIMIDO 5,4-D]PYRIMIDINES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION THOMAE GMBH DR K (DE) 2003-10-15 EP disclosed