SCHEMBL6990971

SCHEMBL6990971

CN(C)CCCn1ccc2ccc(C#N)cc21

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.50
HTR2C P28335 3/20 0.50
HTR1D P28221 9/20 0.48
NOS3 P29474 4/20 0.47
NOS1 P29475 4/20 0.47
BPTF Q12830 1/20 0.45
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
TSHR P16473 3/20 0.44
HSD17B10 Q99714 3/20 0.44
HPGD P15428 2/20 0.44
GLA P06280 1/20 0.44
HTT P42858 1/20 0.44
USP2 O75604 1/20 0.43
POLB P06746 1/20 0.43
NOS2 P35228 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6995071 0.99 HTR2A (0.49) HTR2AHTR2CHTR1DNOS3NOS1
SCHEMBL27400361 0.92 HTR2A (0.59) HTR2AHTR2CHTR1DNOS3NOS1
SCHEMBL6996636 0.86 ALDH1A1 (0.47) HTR2AHTR2CHTR1DNOS3NOS1
SCHEMBL8430655 0.84 ALDH1A1 (0.46) KDM4EALDH1A1TSHRHSD17B10HPGD
SCHEMBL6993894 0.83 ALDH1A1 (0.50) HTR1DKDM4EALDH1A1TSHRHSD17B10
SCHEMBL6990162 0.82 ALDH1A1 (0.51) HTR2AHTR2CHTR1DKDM4EALDH1A1
SCHEMBL9994932 0.81 ALDH1A1 (0.46) KDM4EALDH1A1TSHRHSD17B10HPGD
SCHEMBL6995817 0.81 ALDH1A1 (0.49) KDM4EALDH1A1TSHRHSD17B10HPGD
SCHEMBL8255718 0.81 ALDH1A1 (0.46) KDM4EALDH1A1TSHRHSD17B10HPGD
SCHEMBL8430662 0.81 ALDH1A1 (0.48) HTR2AHTR2CKDM4EALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023898-B1 Cyano-indoles as serotonine reuptake inhibitors and as 5-HT2c receptor ligands SERVIER LAB (FR) 2003-03-12 EP disclosed
US-6239129-B1 CHARACTERISED BY AN INDOLE RING ON THE AROMATIC MOIETY BY A CYANO GROUP AND ON THE INDOLE NITROGEN BY AN AMINOALKYL CHAIN. GREAT AFFINITY FOR 5-HT2C RECEPTORS, USEFUL FOR DEPRESSION, PANIC ATTACKS, OBSESSIVE-COMPULSIVE DISORDERS, PHOBIAS, ADIR ET COMPAGNIE (FR) 2001-05-29 US disclosed
EP-1023898-A1 Cyano-indoles as serotonine reuptake inhibitors and as 5-HT2c receptor ligands ADIR ET COMPAGNIE (FR) 2000-08-02 EP disclosed