Bicarbonate

Bicarbonate

SCHEMBL6992780

COc1ccc(CC(=O)NC2CCCCC2)c(C)c1.O=C(O)O

nearest known ligand 0.73

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.73
KMT2A Q03164 5/20 0.73
EPHX2 P34913 1/20 0.62
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 2/20 0.56
CYP2C19 P33261 2/20 0.56
HPGD P15428 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
MAPT P10636 1/20 0.55
ALDH1A1 P00352 1/20 0.55
APOBEC3A P31941 1/20 0.55
APOBEC3G Q9HC16 1/20 0.55
POLB P06746 2/20 0.53
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
KLF5 Q13887 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL6996071 1.00 MEN1 (0.73) MEN1KMT2AEPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL6990357 0.99 MEN1 (0.71) MEN1KMT2AEPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL6996704 0.89 MEN1 (0.58) MEN1KMT2AEPHX2HPGDSMN1; SMN2
Bicarbonate SCHEMBL6990325 0.88 MEN1 (0.57) MEN1KMT2AEPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL6998215 0.87 MEN1 (0.57) MEN1KMT2AEPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL6996203 0.87 MEN1 (0.56) MEN1KMT2AEPHX2HPGDALDH1A1
Bicarbonate SCHEMBL6998126 0.87 MEN1 (0.56) MEN1KMT2AEPHX2HPGDMAPT
Bicarbonate SCHEMBL4434715 0.86 KMT2A (0.72) MEN1KMT2AEPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL4428096 0.86 KMT2A (0.72) MEN1KMT2AEPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL8796331 0.86 MEN1 (0.55) MEN1KMT2AEPHX2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0754175-B1 ALKOXY-ALKYL-SUBSTITUTED 1-H-3-ARYL-PYRROLIDINE-2,4-DIONES USED AS HERBICIDES AND PESTICIDES BAYER CROPSCIENCE AG (DE) 2003-01-29 EP disclosed
WO-1995026954-A1 ALKOXY-ALKYL-SUBSTITUTED 1-H-3-ARYL-PYRROLIDINE-2,4-DIONES USED AS HERBICIDES AND PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1995-10-12 WO disclosed