SCHEMBL6993357

SCHEMBL6993357

CCC(c1ccc2c(c1)NC(=O)C(C)O2)N(C)c1cccs1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.42
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
SMYD3 Q9H7B4 3/20 0.36
KDR P35968 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
MAOB P27338 1/20 0.33
ADORA2A P29274 1/20 0.33
HSD17B10 Q99714 2/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8113173 0.88 PARP1 (0.48) PARP1PDE3BPDE3ASMYD3KDR
SCHEMBL6998253 0.78 PARP1 (0.54) PARP1PDE3BPDE3ASMYD3KDR
SCHEMBL7711223 0.78 PARP1 (0.38) PARP1PDE3BPDE3ASMYD3KDR
SCHEMBL8104372 0.77
Hydrochloric Acid SCHEMBL6994569 0.76
SCHEMBL8104377 0.76
SCHEMBL6994127 0.73 PARP1 (0.50) PARP1PDE3BPDE3ASMYD3L3MBTL1
SCHEMBL6995045 0.73 PARP1 (0.50) PARP1PDE3BPDE3ASMYD3L3MBTL1
SCHEMBL6998255 0.72 PARP1 (0.45) PARP1PDE3BPDE3ASMYD3KDR
SCHEMBL8113172 0.71 PARP1 (0.54) PARP1PDE3BPDE3ASMYD3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP disclosed
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed