SCHEMBL7711223

SCHEMBL7711223

CCC(c1ccc2c(c1)NC(=O)C(C)O2)N(Cc1cccs1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.38
GAA P10253 2/20 0.35
HTT P42858 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
POLB P06746 1/20 0.34
SMYD3 Q9H7B4 3/20 0.34
TRPM8 Q7Z2W7 2/20 0.33
RIPK1 Q13546 1/20 0.33
KDR P35968 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
ALDH1A1 P00352 2/20 0.32
HTR1A P08908 1/20 0.32
HTR7 P34969 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7089254 0.92 HTT (0.35) GAAHTTNPSR1POLBTRPM8
SCHEMBL7704922 0.87 PARP1 (0.48) PARP1HTTSMYD3PDE3BPDE3A
SCHEMBL7708174 0.82 GAA (0.37) GAAHTTNPSR1POLBTRPM8
SCHEMBL7708180 0.81 HTT (0.34) GAAHTTNPSR1POLBTRPM8
SCHEMBL7088859 0.79 PARP1 (0.37) PARP1HTTPOLBTRPM8ALDH1A1
SCHEMBL7711431 0.78 PARP1 (0.37) PARP1GAASMYD3KDRPDE3B
SCHEMBL6993357 0.78 PARP1 (0.42) PARP1SMYD3KDRPDE3BPDE3A
SCHEMBL7711130 0.76 PARP1 (0.53) PARP1HTTSMYD3PDE3BPDE3A
SCHEMBL7710846 0.72 PARP1 (0.53) PARP1HTTSMYD3PDE3BPDE3A
SCHEMBL7711394 0.72 PARP1 (0.36) PARP1GAASMYD3KDRPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed