SCHEMBL6993773

SCHEMBL6993773

OCc1cccc(Nc2ncnc3cnc(NC4CCC(O)CC4)nc23)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.53
EGFR P00533 12/20 0.49
ERBB2 P04626 1/20 0.49
HPGD P15428 1/20 0.49
HTT P42858 1/20 0.49
SYK P43405 1/20 0.46
MAPK8 P45983 1/20 0.46
MAPK9 P45984 1/20 0.46
GSK3A P49840 1/20 0.45
GSK3B P49841 1/20 0.45
IRAK4 Q9NWZ3 1/20 0.44
CDK1 P06493 2/20 0.43
FLT3 P36888 1/20 0.43
TYRO3 Q06418 1/20 0.43
MERTK Q12866 1/20 0.43
GAS6 Q14393 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993782 1.00 BRAF (0.53) BRAFEGFRERBB2HPGDHTT
SCHEMBL8320282 0.86 CSNK2A1 (0.56) BRAFEGFRERBB2HPGDHTT
SCHEMBL8315969 0.86 EGFR (0.66) BRAFEGFRERBB2HPGDHTT
SCHEMBL8320277 0.86 CSNK2A1 (0.56) BRAFEGFRERBB2HPGDHTT
SCHEMBL8319114 0.86 EGFR (0.67) BRAFEGFRERBB2HPGDHTT
SCHEMBL8316922 0.86 EGFR (0.58) BRAFEGFRERBB2HPGDHTT
SCHEMBL8317438 0.86 EGFR (0.66) BRAFEGFRERBB2HPGDHTT
SCHEMBL8316918 0.86 EGFR (0.58) BRAFEGFRERBB2HPGDHTT
SCHEMBL8319108 0.86 EGFR (0.67) BRAFEGFRERBB2HPGDHTT
SCHEMBL8315961 0.86 EGFR (0.66) BRAFEGFRERBB2HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888351-B1 PYRIMIDO 5,4-D]PYRIMIDINES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION THOMAE GMBH DR K (DE) 2003-10-15 EP disclosed
EP-0888351-A1 PYRIMIDO 5,4-D]PYRIMIDINES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION Dr. Karl Thomae GmbH (DE) 1999-01-07 EP disclosed
WO-1997032880-A1 PYRIMIDO[5,4-D]PYRIMIDINES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION DR. KARL THOMAE GMBH (DE) 1997-09-12 WO disclosed