SCHEMBL6994029

SCHEMBL6994029

Fc1ccc(C23CCCN2CCC3)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 5/20 0.43
GRIN2A Q12879 5/20 0.43
GRIN2B Q13224 5/20 0.43
PRCP P42785 3/20 0.43
KCNH2 Q12809 2/20 0.43
SIGMAR1 Q99720 2/20 0.43
GRIN2D O15399 1/20 0.43
GRIN3B O60391 1/20 0.43
CYP2B6 P20813 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
GRIN2C Q14957 1/20 0.43
GRIN3A Q8TCU5 1/20 0.43
OPRM1 P35372 3/20 0.42
OPRD1 P41143 1/20 0.42
SLC6A9 P48067 5/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6998256 0.98 OPRM1 (0.45) GRIN1GRIN2AGRIN2BPRCPKCNH2
SCHEMBL6991802 0.79 GRIN1 (0.43) GRIN1GRIN2AGRIN2BPRCPKCNH2
SCHEMBL6990087 0.79 GRIN1 (0.45) GRIN1GRIN2AGRIN2BPRCPKCNH2
Hydrochloric Acid SCHEMBL6999479 0.78 OPRM1 (0.45) GRIN1GRIN2AGRIN2BPRCPKCNH2
Hydrochloric Acid SCHEMBL6992181 0.78 OPRM1 (0.45) GRIN1GRIN2AGRIN2BPRCPKCNH2
SCHEMBL6997844 0.72 GRIN1 (0.37) GRIN1GRIN2AGRIN2BPRCPKCNH2
SCHEMBL6995444 0.72 GRIN1 (0.37) GRIN1GRIN2AGRIN2BPRCPKCNH2
SCHEMBL6992209 0.72 GRIN1 (0.37) GRIN1GRIN2AGRIN2BPRCPKCNH2
Hydrochloric Acid SCHEMBL7001900 0.71 OPRM1 (0.38) GRIN1GRIN2AGRIN2BPRCPKCNH2
Hydrochloric Acid SCHEMBL7001597 0.71 OPRM1 (0.38) GRIN1GRIN2AGRIN2BPRCPKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970083-B1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2003-04-16 EP claimed
EP-0970083-A1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-01-12 EP claimed
WO-1998037082-A1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1998-08-27 WO claimed
WO-2008049554-A1 USE OF 7A-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS FOR CONTROLLING ANIMAL PESTS BAYER CROPSCIENCE AG (DE) 2008-05-02 WO disclosed
EP-0970083-B1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2003-04-16 EP disclosed
EP-0970083-A1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-01-12 EP disclosed
WO-1998037082-A1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1998-08-27 WO disclosed
US-5733912-A NERVOUS SYSTEM DISORDERS IN NERVE CELLS ABBOTT LABORATORIES (US) 1998-03-31 US disclosed