SCHEMBL6994458

SCHEMBL6994458

Oc1ccc2cc(COc3ccccc3)ccc2c1C1=NCCc2ccccc21

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.34
MAOB P27338 3/20 0.34
GRM5 P41594 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
S1PR1 P21453 1/20 0.34
FFAR1 O14842 1/20 0.33
RAB9A P51151 1/20 0.33
CMKLR1 Q99788 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
HSD17B1 P14061 1/20 0.33
CYP2B6 P20813 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B2 P37059 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983448 0.78 MAOA (0.39) MAOAESR1ESR2RAB9ACYP1A2
SCHEMBL6985896 0.77 MAOA (0.44) MAOACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6992467 0.74 MAOA (0.48) MAOACYP3A4
SCHEMBL6986780 0.72 MAOA (0.40) MAOARAB9A
SCHEMBL6716154 0.70 GSTP1 (0.48) MAOAMAOBRAB9ACYP1A2CYP2C19
SCHEMBL6986039 0.66 GAA (0.41) MAOAESR1RAB9ACYP1A2
SCHEMBL6986047 0.66 MAOA (0.43) MAOARAB9A
SCHEMBL13651006 0.66 MAOA (0.60) MAOA
SCHEMBL6986057 0.66 MAOA (0.40) MAOAESR1ESR2CYP3A4
SCHEMBL6983460 0.65 MAOA (0.39) MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183378-B2 Ligands, their preparation and uses thereof in asymmetric reactions Li, Chao-Jun (CA) 2012-05-22 US disclosed