SCHEMBL6994580

SCHEMBL6994580

COc1ccc2c(c1OC)C[C@H](C1CCN(S(C)(=O)=O)CC1)O[C@@H]2CN

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.43
ADRA2B P18089 2/20 0.43
ADRA2C P18825 2/20 0.43
HTR2C P28335 2/20 0.43
SLC6A3 Q01959 2/20 0.43
DRD1 P21728 3/20 0.43
PARP1 P09874 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 2/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 2/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994578 1.00 ADRA2A (0.43) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL6994586 1.00 ADRA2A (0.43) ADRA2AADRA2BADRA2CHTR2CSLC6A3
Hydrochloric Acid SCHEMBL6996332 0.99 ADRA2A (0.43) ADRA2AADRA2BADRA2CHTR2CSLC6A3
Hydrochloric Acid SCHEMBL6996329 0.99 ADRA2A (0.43) ADRA2AADRA2BADRA2CHTR2CSLC6A3
Hydrochloric Acid SCHEMBL6996335 0.99 ADRA2A (0.43) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL6988766 0.85 DRD1 (0.38) DRD1PARP1SMN1; SMN2TSHRGAA
SCHEMBL6988760 0.85 DRD1 (0.38) DRD1PARP1SMN1; SMN2TSHRGAA
SCHEMBL6988755 0.85 DRD1 (0.38) DRD1PARP1SMN1; SMN2TSHRGAA
SCHEMBL6998208 0.85 ADRA2A (0.45) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL6998213 0.85 ADRA2A (0.45) ADRA2AADRA2BADRA2CHTR2CSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015446-B1 (4-PIPERIDINYL)-1H-2-BENZOPYRAN DERIVATIVES USEFUL AS ANTIPSYCHOTIC AGENTS AVENTIS PHARMA INC (US) 2003-04-02 EP claimed
US-6004982-A SIDE EFFECT REDUCTION; SCHIZOPHRENIA HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US claimed
EP-1015446-B1 (4-PIPERIDINYL)-1H-2-BENZOPYRAN DERIVATIVES USEFUL AS ANTIPSYCHOTIC AGENTS AVENTIS PHARMA INC (US) 2003-04-02 EP disclosed
US-6004982-A SIDE EFFECT REDUCTION; SCHIZOPHRENIA HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed