SCHEMBL6996957

SCHEMBL6996957

CC1=C(N)Nc2cc(CN(C)c3ccncc3)ccc2O1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.36
HDAC3 O15379 1/20 0.36
NR3C2 P08235 1/20 0.34
EGFR P00533 1/20 0.32
CSF1R P07333 1/20 0.32
HIF1A Q16665 2/20 0.31
EPAS1 Q99814 2/20 0.31
TYMS P04818 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6991853 0.99 HDAC1 (0.35) HDAC1HDAC3NR3C2EGFRCSF1R
Hydrochloric Acid SCHEMBL7001589 0.87 GBA1 (0.36) NR3C2EGFRCSF1RHIF1AEPAS1
Hydrochloric Acid SCHEMBL6995850 0.82 NR3C2 (0.33) NR3C2
SCHEMBL7001780 0.80 NR3C2 (0.34) NR3C2
Hydrochloric Acid SCHEMBL6988645 0.79 NR3C2 (0.33) NR3C2
Hydrochloric Acid SCHEMBL6992156 0.78 NR3C2 (0.33) NR3C2HIF1AEPAS1
SCHEMBL6989624 0.74 PARP1 (0.52) HDAC1NR3C2
SCHEMBL6999827 0.73 NOS1 (0.46)
SCHEMBL7000588 0.71 PARP1 (0.37)
Hydrochloric Acid SCHEMBL6999676 0.68 PARP1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed