SCHEMBL6997064

SCHEMBL6997064

CSc1ccc(C2=C(c3ccccc3)C(=O)OC23CCCC3)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.54
PTGS1 P23219 7/20 0.52
GSK3B P49841 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
EDNRA P25101 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997168 0.97 PTGS2 (0.54) PTGS2PTGS1GSK3BSMN1; SMN2KDM4E
SCHEMBL6991312 0.80 PTGS2 (0.64) PTGS2PTGS1ALDH1A1
SCHEMBL6993378 0.77 PTGS2 (0.64) PTGS2PTGS1ALDH1A1
SCHEMBL6986739 0.77 PTGS2 (0.54) PTGS2PTGS1ALDH1A1HPGD
SCHEMBL6988455 0.76 PTGS2 (0.52) PTGS2PTGS1ALDH1A1HPGD
SCHEMBL8799520 0.76 PTGS2 (0.52) PTGS2PTGS1ALDH1A1HPGD
SCHEMBL8799123 0.76 PTGS2 (0.52) PTGS2PTGS1ALDH1A1HPGD
SCHEMBL6989032 0.75 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL6989030 0.74 PTGS2 (0.67) PTGS2PTGS1ALDH1A1
SCHEMBL7573008 0.71 PTGS2 (0.57) PTGS2PTGS1GSK3BSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799218-B1 DIARYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2003-02-19 EP disclosed
US-6222048-B1 AS ANTIINFLAMMATORY, ANTIPYRETIC AND ANALGESIC AGENTS; INHIBITS HORMONE INDUCED UTERINE CONTRACTION; ANTICANCER PROPERTIES; SIDE EFFECT REDUCTION MERCK FROSST CANADA & CO. (CA) 2001-04-24 US disclosed
WO-1996019469-A1 DIARYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1996-06-27 WO disclosed