SCHEMBL6997437

SCHEMBL6997437

c1ccc(-c2cncc(C34CCCN3CCC4)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.50
GRIN1 Q05586 2/20 0.50
GRIN2A Q12879 2/20 0.50
GRIN2B Q13224 2/20 0.50
SLC6A3 Q01959 2/20 0.50
GRIN2D O15399 1/20 0.50
GRIN3B O60391 1/20 0.50
CYP2B6 P20813 1/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A4 P31645 1/20 0.50
PRCP P42785 1/20 0.50
KCNH2 Q12809 1/20 0.50
GRIN2C Q14957 1/20 0.50
GRIN3A Q8TCU5 1/20 0.50
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49
CHRNA7 P36544 1/20 0.40
CYP11B2 P19099 1/20 0.39
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6999017 0.98 OPRM1 (0.51) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
SCHEMBL6994482 0.74 GRIN1 (0.40) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
SCHEMBL6992429 0.74 GRIN1 (0.40) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
SCHEMBL6998974 0.74 GRIN1 (0.40) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
SCHEMBL6995762 0.74 GRIN1 (0.40) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
SCHEMBL6992113 0.74 GRIN1 (0.42) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
Hydrochloric Acid SCHEMBL6997379 0.73 OPRM1 (0.41) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
Hydrochloric Acid SCHEMBL6993575 0.73 OPRM1 (0.41) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
Hydrochloric Acid SCHEMBL6999005 0.73 OPRM1 (0.41) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
Hydrochloric Acid SCHEMBL6995633 0.73 OPRM1 (0.41) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970083-B1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2003-04-16 EP claimed
EP-0970083-B1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2003-04-16 EP disclosed
EP-0970083-A1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-01-12 EP disclosed
WO-1998037082-A1 7a-HETEROCYCLE-SUBSTITUTED HEXAHYDRO-1H-PYRROLIZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1998-08-27 WO disclosed
US-5733912-A NERVOUS SYSTEM DISORDERS IN NERVE CELLS ABBOTT LABORATORIES (US) 1998-03-31 US disclosed