SCHEMBL6997540

SCHEMBL6997540

CC1Oc2ccc(C(N)C(=O)OC(C)(C)C(C)c3ccco3)cc2NC1=O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 3/20 0.38
PARP1 P09874 7/20 0.38
PDE3B Q13370 2/20 0.35
PDE3A Q14432 2/20 0.35
HTR1A P08908 2/20 0.33
HTR7 P34969 2/20 0.33
KDR P35968 1/20 0.32
USP2 O75604 1/20 0.31
GAA P10253 1/20 0.31
KCNH2 Q12809 1/20 0.31
MAOB P27338 1/20 0.30
ADORA2A P29274 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7000031 0.85 SMYD3 (0.38) SMYD3PARP1PDE3BPDE3AHTR1A
SCHEMBL6991325 0.84 SMYD3 (0.36) SMYD3PARP1PDE3BPDE3AHTR1A
SCHEMBL6998315 0.83 SMYD3 (0.37) SMYD3PARP1PDE3BPDE3AHTR1A
SCHEMBL6996791 0.81 CYP2C19 (0.32)
SCHEMBL6998308 0.79 PARP1 (0.46) SMYD3PARP1PDE3BPDE3AHTR1A
SCHEMBL6997632 0.76 PARP1 (0.42) SMYD3PARP1PDE3BPDE3AHTR1A
SCHEMBL7711412 0.75 PARP1 (0.39) SMYD3PARP1PDE3BPDE3AHTR1A
SCHEMBL7000925 0.75 PARP1 (0.42) SMYD3PARP1USP2GAA
SCHEMBL6991269 0.74 PARP1 (0.40) SMYD3PARP1PDE3BPDE3AHTR1A
SCHEMBL6998306 0.74 PARP1 (0.40) SMYD3PARP1PDE3BPDE3AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP disclosed