SCHEMBL6997941

SCHEMBL6997941

CN1CCC(O)(c2ccc3[nH]cc(C4=CCN5CCC[C@@H]5C4)c3c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.41
NOS1 P29475 4/20 0.39
NOS3 P29474 2/20 0.38
NOS2 P35228 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997685 0.91 SLC6A4 (0.36) SLC6A4NOS1NOS3NOS2
SCHEMBL7002561 0.91 SLC6A4 (0.36) SLC6A4NOS1NOS3NOS2
SCHEMBL6999590 0.89 SLC6A4 (0.35) SLC6A4NOS1NOS3NOS2
SCHEMBL7006099 0.81 SLC6A4 (0.53) SLC6A4NOS1NOS3NOS2
SCHEMBL7010984 0.81 SLC6A4 (0.53) SLC6A4NOS1NOS3NOS2
SCHEMBL6999444 0.81 SLC6A4 (0.56) SLC6A4
SCHEMBL6999439 0.81 SLC6A4 (0.56) SLC6A4
SCHEMBL6965518 0.80 SLC6A4 (0.65) SLC6A4
SCHEMBL1122232 0.78 HTR1D (0.43) SLC6A4NOS1NOS3NOS2
SCHEMBL6994351 0.78 SLC6A4 (0.56) SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562809-B1 Contraction of coronary arteries may be mediated by its stimulation of the 5-HT1B (formerly 5-HT1D beta); compounds selective for a 5-HT1D receptor NPS ALLELIX CORP. (CA) 2003-05-13 US claimed
EP-1114049-B1 3-BICYCLOINDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-03-19 EP claimed
US-6562809-B1 Contraction of coronary arteries may be mediated by its stimulation of the 5-HT1B (formerly 5-HT1D beta); compounds selective for a 5-HT1D receptor NPS ALLELIX CORP. (CA) 2003-05-13 US disclosed
EP-1114049-B1 3-BICYCLOINDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-03-19 EP disclosed
EP-1114049-A1 3-BICYCLOINDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS Allelix Corp. (CA) 2001-07-11 EP disclosed
WO-2000017198-A1 3-BICYCLOINDOLE COMPOUNDS AS 5-HT1D LIGANDS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-03-30 WO disclosed