SCHEMBL6998092

SCHEMBL6998092

CNCC1OC(C2CCN(CCc3ccc(F)cc3)CC2)Cc2c1ccc(OC)c2OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.51
GRM2 Q14416 3/20 0.51
DRD1 P21728 5/20 0.49
HTR2C P28335 4/20 0.49
HRH1 P35367 4/20 0.49
ADRA1B P35368 4/20 0.49
HTR2B P41595 4/20 0.49
DRD2 P14416 3/20 0.49
ADRA2B P18089 1/20 0.49
OPRK1 P41145 1/20 0.49
KCNQ1 P51787 1/20 0.49
KCNH2 Q12809 1/20 0.49
TMEM97 Q5BJF2 1/20 0.49
DRD4 P21917 3/20 0.43
HRH2 P25021 3/20 0.43
HTR1D P28221 3/20 0.43
HTR1B P28222 3/20 0.43
SLC6A4 P31645 3/20 0.43
HTR7 P34969 3/20 0.43
ADRA2C P18825 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998747 0.91 DRD1 (0.43) HTR2AGRM2DRD1ADRA1BTMEM97
SCHEMBL6998755 0.91 DRD1 (0.43) HTR2AGRM2DRD1ADRA1BTMEM97
SCHEMBL6998751 0.91 DRD1 (0.43) HTR2AGRM2DRD1ADRA1BTMEM97
SCHEMBL7001096 0.90 HTR2A (0.49) HTR2AGRM2DRD1HTR2CHRH1
SCHEMBL6992748 0.84 DRD1 (0.63) HTR2AGRM2DRD1ADRA1BADRA2B
Bromide SCHEMBL6998756 0.83 DRD1 (0.62) HTR2AGRM2DRD1ADRA1BADRA2B
SCHEMBL6992458 0.82 DRD1 (0.42) HTR2AGRM2DRD1HTR2CHRH1
SCHEMBL6998880 0.82 DRD1 (0.41) HTR2AGRM2DRD1ADRA1BTMEM97
SCHEMBL6998873 0.82 DRD1 (0.41) HTR2AGRM2DRD1ADRA1BTMEM97
SCHEMBL6998889 0.82 DRD1 (0.41) HTR2AGRM2DRD1ADRA1BTMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015446-B1 (4-PIPERIDINYL)-1H-2-BENZOPYRAN DERIVATIVES USEFUL AS ANTIPSYCHOTIC AGENTS AVENTIS PHARMA INC (US) 2003-04-02 EP disclosed
US-6004982-A SIDE EFFECT REDUCTION; SCHIZOPHRENIA HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed