SCHEMBL7003085

SCHEMBL7003085

C1=C(c2c[nH]c3ccc(OC4CCCCC4)cc23)C[C@H]2CCCN2C1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.48
SLC6A4 P31645 3/20 0.44
HTR1A P08908 4/20 0.40
DRD2 P14416 4/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
HTR1D P28221 1/20 0.39
HTR2C P28335 1/20 0.39
MAPK1 P28482 1/20 0.39
BRCA1 P38398 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7003088 1.00 HTR6 (0.48) HTR6SLC6A4HTR1ADRD2ALDH1A1
SCHEMBL6994448 0.87 SLC6A4 (0.59) HTR6SLC6A4HTR1ADRD2ALDH1A1
SCHEMBL6994454 0.87 SLC6A4 (0.59) HTR6SLC6A4HTR1ADRD2ALDH1A1
SCHEMBL1122232 0.85 HTR1D (0.43) SLC6A4HTR1D
SCHEMBL6998384 0.84 JAK2 (0.47) HTR6SLC6A4HTR1ADRD2ALDH1A1
SCHEMBL6999444 0.82 SLC6A4 (0.56) SLC6A4HTR1D
SCHEMBL6999439 0.82 SLC6A4 (0.56) SLC6A4HTR1D
SCHEMBL6994351 0.81 SLC6A4 (0.56) HTR6SLC6A4HTR1ADRD2HTR2C
SCHEMBL6641862 0.81 SLC6A4 (0.56) HTR6SLC6A4HTR1ADRD2HTR2A
SCHEMBL6996253 0.81 SLC6A4 (0.56) HTR6SLC6A4HTR1ADRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562809-B1 Contraction of coronary arteries may be mediated by its stimulation of the 5-HT1B (formerly 5-HT1D beta); compounds selective for a 5-HT1D receptor NPS ALLELIX CORP. (CA) 2003-05-13 US claimed
EP-1114049-B1 3-BICYCLOINDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-03-19 EP claimed
US-6562809-B1 Contraction of coronary arteries may be mediated by its stimulation of the 5-HT1B (formerly 5-HT1D beta); compounds selective for a 5-HT1D receptor NPS ALLELIX CORP. (CA) 2003-05-13 US disclosed
EP-1114049-B1 3-BICYCLOINDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-03-19 EP disclosed