SCHEMBL7003678

SCHEMBL7003678

CC1(C)OC(c2ccc(S(N)(=O)=O)cc2Cl)=C(c2cccc(F)c2)C1=O

nearest known ligand 0.73

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.47
PTGS1 P23219 10/20 0.47
CA4 P22748 2/20 0.42
BRAF P15056 1/20 0.40
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
CA13 Q8N1Q1 1/20 0.38
CA12 O43570 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
PGR P06401 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6999969 0.91 PTGS2 (0.55) PTGS2PTGS1BRAF
SCHEMBL7001135 0.90 PTGS2 (0.39) PTGS2PTGS1CA4BRAFCA1
SCHEMBL7001723 0.89 PTGS2 (0.48) PTGS2PTGS1CA4BRAFCA1
SCHEMBL7001112 0.89 CA1 (0.43) PTGS2PTGS1CA4CA1CA2
SCHEMBL7001070 0.88 PTGS2 (0.41) PTGS2PTGS1CA4CA1CA2
SCHEMBL7003146 0.88 PTGS2 (0.42) PTGS2PTGS1CA4CA1CA2
Polmacoxib SCHEMBL3233093 0.85 PTGS2 (0.55) PTGS2PTGS1CA1CA2CA9
Polmacoxib SCHEMBL29351757 0.85 PTGS2 (0.55) PTGS2PTGS1CA1CA2CA9
SCHEMBL7002269 0.84 BRAF (0.41) PTGS2PTGS1CA4BRAFCA1
SCHEMBL6997219 0.83 CA1 (0.41) PTGS2PTGS1CA4BRAFCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP claimed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US claimed
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP disclosed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US disclosed