SCHEMBL700400

SCHEMBL700400

COc1cccc(NC2CCN(c3nc(-c4ccncc4F)cc(=O)n3C)C2)c1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 18/20 0.53
CYP2D6 P10635 8/20 0.53
CYP1A2 P05177 3/20 0.53
ROCK2 O75116 2/20 0.51
CYP3A4 P08684 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL697459 1.00 GSK3B (0.53) GSK3BCYP2D6CYP1A2ROCK2CYP3A4
SCHEMBL88507 0.95 ROCK2 (0.53) GSK3BCYP2D6CYP1A2ROCK2CYP3A4
SCHEMBL8232344 0.86 GSK3B (0.62) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL695308 0.86 GSK3B (0.62) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL699010 0.86 GSK3B (0.54) GSK3BCYP2D6CYP1A2
SCHEMBL88156 0.85 GSK3B (0.51) GSK3BCYP2D6CYP1A2ROCK2CYP3A4
SCHEMBL698073 0.85 GSK3B (0.64) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL8235419 0.85 GSK3B (0.64) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL87814 0.82 GSK3B (0.49) GSK3BCYP2D6CYP1A2ROCK2
SCHEMBL8344265 0.81 GSK3B (0.59) GSK3BCYP2D6CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423207-A2 2-(cyclic amino)-pyrimidone derivatives as TPK1 inhibitors Mitsubishi Tanabe Pharma Corporation (JP) 2012-02-29 EP disclosed