SCHEMBL7004146

SCHEMBL7004146

c1ccc2c(CCCCc3c[nH]c4ccccc34)c[nH]c2c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.71
CYP3A4 P08684 2/20 0.71
HTR2C P28335 2/20 0.71
HTR6 P50406 2/20 0.71
MPO P05164 1/20 0.71
CYP1A2 P05177 1/20 0.71
CYP2D6 P10635 1/20 0.71
CYP2A6 P11509 1/20 0.71
NFKB1 P19838 1/20 0.71
HTR1D P28221 1/20 0.71
HTR1B P28222 1/20 0.71
HTR7 P34969 1/20 0.71
CTSK P43235 1/20 0.71
CYP2A13 Q16696 1/20 0.71
TAAR1 Q96RJ0 1/20 0.71
SLC6A4 P31645 2/20 0.71
MAPT P10636 2/20 0.69
TDP1 Q9NUW8 2/20 0.69
MEN1 O00255 1/20 0.69
AHR P35869 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7001306 0.98 HTR2A (0.69) HTR2ACYP3A4HTR2CHTR6MPO
SCHEMBL7889427 0.98 HTR2A (0.69) HTR2ACYP3A4HTR2CHTR6MPO
SCHEMBL7004071 0.98 HTR2A (0.69) HTR2ACYP3A4HTR2CHTR6MPO
SCHEMBL7005718 0.96 HTR2A (0.71) HTR2ACYP3A4HTR2CHTR6MPO
SCHEMBL4985934 0.91 HTR2A (0.77) HTR2ACYP3A4HTR2CHTR6MPO
SCHEMBL109955 0.91 SLC6A4 (0.66) HTR2ACYP3A4HTR2CHTR6MPO
SCHEMBL734204 0.91 SLC6A4 (0.61) HTR2ACYP3A4HTR2CHTR6MPO
SCHEMBL7495793 0.91 SLC6A4 (0.61) HTR2ACYP3A4HTR2CHTR6MPO
SCHEMBL4636791 0.91 SLC6A4 (0.61) HTR2ACYP3A4HTR2CHTR6MPO
SCHEMBL7280016 0.91 SLC6A4 (0.61) HTR2ACYP3A4HTR2CHTR6MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337511-A1 BIS-HETEROCYCLIC COMPOUNDS WITH ANTITUMOUR AND CHEMOSENSITISING ACTIVITY Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 2003-08-27 EP disclosed
WO-2002036561-A1 BIS-HETEROCYCLIC COMPOUNDS WITH ANTITUMOUR AND CHEMOSENSITISING ACTIVITY SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2002-05-10 WO disclosed