SCHEMBL7004716

SCHEMBL7004716

CCCCOc1c(CCNC(=O)OC(C)(C)C)n(CC(C)(C)C)c(=O)c2ccc(/C=C/C(=O)O)cc12

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2B6 P20813 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP3A43 Q9HB55 1/20 0.38
AKR1C3 P42330 1/20 0.36
ESR1 P03372 7/20 0.34
ESR2 Q92731 6/20 0.34
KDM4E B2RXH2 1/20 0.34
DYRK1A Q13627 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RXRA P19793 1/20 0.33
DPP4 P27487 1/20 0.33
CNR2 P34972 1/20 0.33
POLB P06746 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236103 0.92 CYP1A1 (0.36) CYP1A1CYP2D6CYP2B6CYP2C19CYP3A43
SCHEMBL5236095 0.92 CYP1A1 (0.36) CYP1A1CYP2D6CYP2B6CYP2C19CYP3A43
SCHEMBL5236373 0.85 DPP4 (0.40) CYP1A1CYP2D6CYP2B6CYP2C19CYP3A43
SCHEMBL5236382 0.85 DPP4 (0.40) CYP1A1CYP2D6CYP2B6CYP2C19CYP3A43
SCHEMBL5238832 0.83 DPP4 (0.43) CYP1A1CYP2D6CYP2B6CYP2C19CYP3A43
SCHEMBL5238822 0.83 DPP4 (0.43) CYP1A1CYP2D6CYP2B6CYP2C19CYP3A43
SCHEMBL5232143 0.77 KDM4E (0.37) CYP1A1CYP2D6CYP2B6CYP2C19CYP3A43
SCHEMBL7564209 0.77 DPP4 (0.50) ESR1ESR2KDM4EDPP4
Hydrochloric Acid SCHEMBL5237626 0.76 DPP4 (0.51) ESR1ESR2KDM4EDPP4
Hydrochloric Acid SCHEMBL5237614 0.76 DPP4 (0.51) ESR1ESR2KDM4EDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed