SCHEMBL7004969

SCHEMBL7004969

Nc1cc(-n2cc(C(=O)O)c(=O)c3cc(F)c(N4CC[C@H](N)C4)c(Cl)c32)c(F)cc1F

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.69
POLB P06746 1/20 0.69
CHRM2 P08172 1/20 0.69
CHRM1 P11229 1/20 0.69
OPRM1 P35372 1/20 0.69
OPRD1 P41143 1/20 0.69
TOP2A P11388 15/20 0.62
TOP1 P11387 3/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2C9 P11712 1/20 0.62
TOP2B Q02880 10/20 0.62
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8479016 1.00 ALDH1A1 (0.69) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7010026 1.00 ALDH1A1 (0.69) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL8482368 0.94 ALDH1A1 (0.68) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7014529 0.94 ALDH1A1 (0.68) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7004804 0.93 CYP3A4 (0.71) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7013670 0.91 TOP2A (0.64) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL19728359 0.91 ALDH1A1 (0.64) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7012041 0.89 KCNH2 (0.56) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL8482489 0.89 TOP2A (0.57) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7004713 0.89 TOP2A (0.57) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787720-B1 PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KK (JP) 2003-07-16 EP disclosed
US-5910498-A NOVEL COMPOUNDS HAVING REDUCED CYTOTOXICITY, PHOTOTOXICITY; TREATING BACTERIAL AND VIRAL INFECTIONS WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1999-06-08 US disclosed
EP-0787720-A1 NOVEL PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1997-08-06 EP disclosed