SCHEMBL7005138

SCHEMBL7005138

O=COCc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.45
ERN1 O75460 1/20 0.39
IDO1 P14902 2/20 0.39
TSHR P16473 3/20 0.39
LMNA P02545 2/20 0.39
VCAM1 P19320 1/20 0.38
CYP3A4 P08684 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
ALOX5 P09917 1/20 0.36
AKR1C3 P42330 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12908868 0.88 ERN1 (0.38) CYP19A1ERN1IDO1TSHRLMNA
SCHEMBL12908867 0.84 TP53 (0.44) LMNACYP3A4SMN1; SMN2ALDH1A1POLB
SCHEMBL12908866 0.83 ALDH1A1 (0.45) TSHRLMNACYP3A4SMN1; SMN2ALDH1A1
SCHEMBL96364 0.82 TSHR (0.57) TSHRLMNASMN1; SMN2ALDH1A1
SCHEMBL1212 0.81 IDO1 (0.61) IDO1TSHRLMNASMN1; SMN2ALDH1A1
SCHEMBL96621 0.78 ALDH1A1 (0.42) CYP19A1TSHRCYP3A4SMN1; SMN2ALDH1A1
SCHEMBL11273785 0.78 CYP19A1 (0.50) CYP19A1IDO1TSHRLMNAVCAM1
SCHEMBL9808020 0.76 CYP19A1 (0.48) CYP19A1IDO1TSHRLMNAVCAM1
SCHEMBL535425 0.76 IDO1 (0.66) CYP19A1IDO1TSHRLMNAVCAM1
SCHEMBL19766404 0.75 CYP19A1 (0.52) CYP19A1ERN1TSHRLMNAVCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108430998-B Azabicyclo derivatives, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-07-09 CN disclosed
EP-1081149-B1 PYRAZOLO 1,5-a]PYRIMIDINE DERIVATIVES OTSUKA PHARMA CO LTD (JP) 2003-04-02 EP disclosed
US-6372749-B1 PHARMACOLOGICAL EFFECTS SUCH AS ANALGESIC ACTION, INHIBITORY EFFECT ON NITROGEN MONOXIDE SYNTHETASE AND THE LIKE AND ARE USEFUL AS ANALGESICS. OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2002-04-16 US disclosed
EP-1081149-A1 PYRAZOLO 1,5-a]PYRIMIDINE DERIVATIVES OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2001-03-07 EP disclosed