SCHEMBL7005568

SCHEMBL7005568

Cc1nnc(-c2cc3c(Nc4ccc(S(=O)(=O)c5ccccc5)cc4)ncnc3cn2)o1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.45
ERBB2 P04626 5/20 0.45
MAPK1 P28482 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HTT P42858 1/20 0.42
BRAF P15056 1/20 0.41
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
HIF1A Q16665 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
LRRK2 Q5S007 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PIP4K2A P48426 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005581 0.87 EGFR (0.37) EGFRERBB2MAPK1KDM4EHTT
SCHEMBL6773317 0.85 BRAF (0.53) EGFRERBB2MAPK1KDM4EHTT
Hydrochloric Acid SCHEMBL6768785 0.85 BRAF (0.52) EGFRERBB2MAPK1KDM4EHTT
SCHEMBL7010037 0.84 EGFR (0.55) EGFRERBB2MAPK1KDM4EHTT
SCHEMBL7008227 0.81 ERBB2 (0.65) EGFRERBB2CLK4
SCHEMBL7890444 0.79 EGFR (0.47) EGFRERBB2MAPK1KDM4EHTT
SCHEMBL3321532 0.78 EGFR (0.51) EGFRERBB2MAPK1KDM4EHTT
Hydrochloric Acid SCHEMBL3320236 0.77 EGFR (0.50) EGFRERBB2MAPK1KDM4EHTT
SCHEMBL3320152 0.77 ERBB2 (0.58) EGFRERBB2BRAFHSD17B10
SCHEMBL3324098 0.77 EGFR (0.57) EGFRERBB2MAPK1KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912572-B1 BICYCLIC HETEROAROMATIC COMPOUNDS AS PROTEIN TYROSINE KINASE INHIBITORS GLAXO GROUP LTD (GB) 2003-01-15 EP disclosed