SCHEMBL7010037

SCHEMBL7010037

Cc1nnc(-c2cc3c(Nc4ccc(Oc5ccccc5)cc4)ncnc3cn2)o1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.55
RIPK2 O43353 1/20 0.55
EPHB2 P29323 1/20 0.55
KDR P35968 1/20 0.54
TEK Q02763 1/20 0.54
ERBB2 P04626 8/20 0.50
ERBB4 Q15303 3/20 0.48
JAK3 P52333 2/20 0.48
TTBK1 Q5TCY1 1/20 0.46
TTBK2 Q6IQ55 1/20 0.46
MAPT P10636 3/20 0.46
TP53 P04637 2/20 0.46
LMNA P02545 1/20 0.45
KDM4E B2RXH2 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
GRM1 Q13255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7008227 0.89 ERBB2 (0.65) EGFRERBB2ERBB4TTBK1TTBK2
SCHEMBL6764388 0.85 KDR (0.58) EGFRRIPK2EPHB2KDRTEK
SCHEMBL7005568 0.84 EGFR (0.45) EGFRKDRERBB2LMNAKDM4E
Hydrochloric Acid SCHEMBL6766661 0.84 KDR (0.57) EGFRRIPK2EPHB2KDRTEK
SCHEMBL7009435 0.81 EGFR (0.58) EGFRERBB2ERBB4JAK3
SCHEMBL6769401 0.76 ERBB2 (0.67) EGFRERBB2ERBB4JAK3MAPT
SCHEMBL7888611 0.76 KDR (0.66) EGFRRIPK2EPHB2KDRTEK
SCHEMBL16981193 0.76 EGFR (0.73) EGFRRIPK2EPHB2KDRTEK
SCHEMBL7886379 0.76 EGFR (0.63) EGFRRIPK2EPHB2KDRTEK
Hydrochloric Acid SCHEMBL6769685 0.75 ERBB2 (0.66) EGFRERBB2ERBB4JAK3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912572-B1 BICYCLIC HETEROAROMATIC COMPOUNDS AS PROTEIN TYROSINE KINASE INHIBITORS GLAXO GROUP LTD (GB) 2003-01-15 EP disclosed