SCHEMBL7005596

SCHEMBL7005596

Clc1cccc([CH]C(Br)c2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.46
MAOB P27338 2/20 0.42
ACP3 P15309 1/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2C9 P11712 1/20 0.41
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
FBP1 P09467 2/20 0.39
CHAT P28329 1/20 0.39
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38
GRIN1 Q05586 3/20 0.38
GRIN2B Q13224 3/20 0.38
GRIN2D O15399 2/20 0.38
GRIN3B O60391 2/20 0.38
GRIN2A Q12879 2/20 0.38
GRIN2C Q14957 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6553126 0.80 ALDH1A1 (0.43) MAOBCYP1A2ALDH1A1CYP2D6
SCHEMBL7008999 0.79 IDO1 (0.47) MAOBCYP1A2IDO1TDO2MAPT
SCHEMBL18243444 0.72 CHRM5 (0.52) CHRM5MAOBCYP1A2CYP2C9FBP1
SCHEMBL7521832 0.72 ACP3 (0.50) ACP3IDO1TDO2KMT2AALDH1A1
Benzaldehyde SCHEMBL20557183 0.72 ALDH1A1 (0.61) CHRM5MAOBCYP1A2CYP2C9FBP1
SCHEMBL23457219 0.72 CHRM5 (0.52) CHRM5MAOBCYP1A2CYP2C9FBP1
SCHEMBL3301775 0.71 CHRM5 (0.56) CHRM5MAOBCYP1A2CYP2C9FBP1
SCHEMBL699875 0.71 CHAT (0.66) CHRM5MAOBCYP1A2CYP2C9FBP1
SCHEMBL29446280 0.71 CHAT (0.66) CHRM5MAOBCYP1A2CYP2C9FBP1
SCHEMBL699874 0.71 CHAT (0.66) CHRM5MAOBCYP1A2CYP2C9FBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1267906-A1 LACTAMS AS INHIBITORS OF A-BETA PROTEIN PRODUCTION Bristol-Myers Squibb Pharma Company (US) 2003-01-02 EP claimed
WO-2001072324-A1 LACTAMS AS INHIBITORS OF A-BETA PROTEIN PRODUCTION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-10-04 WO claimed