SCHEMBL7006936

SCHEMBL7006936

CCOC(=O)c1cn(-c2ccc(F)c(OC)c2)c2c(Cl)c(F)c(F)cc2c1=O

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.56
STAT3 P40763 3/20 0.51
CMA1 P23946 2/20 0.47
NPC1 O15118 1/20 0.44
KDM4E B2RXH2 2/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 2/20 0.41
POLB P06746 1/20 0.41
HSP90AA1 P07900 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
PIM1 P11309 1/20 0.40
ADRB2 P07550 1/20 0.39
THRB P10828 1/20 0.39
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7009901 0.92 HTT (0.57) HTTSTAT3CMA1NPC1KDM4E
SCHEMBL7005983 0.88 HTT (0.56) HTTSTAT3NPC1KDM4EHPGD
SCHEMBL7004828 0.87 ALDH1A1 (0.51) HTTCMA1KDM4EHPGDLMNA
SCHEMBL5528631 0.85 HTT (0.53) HTTSTAT3NPC1KDM4EHPGD
SCHEMBL9871156 0.85 HTT (0.62) HTTSTAT3NPC1KDM4EHPGD
SCHEMBL7005352 0.85 STAT3 (0.51) HTTSTAT3CMA1NPC1KDM4E
SCHEMBL14417317 0.85 HTT (0.52) HTTSTAT3NPC1KDM4EHPGD
SCHEMBL8183513 0.85 HTT (0.57) HTTSTAT3CMA1NPC1KDM4E
SCHEMBL7011166 0.84 NPC1 (0.56) HTTSTAT3CMA1NPC1KDM4E
SCHEMBL5526055 0.83 STAT3 (0.49) HTTSTAT3CMA1NPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0945435-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed