SCHEMBL7006962

SCHEMBL7006962

Cc1cccc(Oc2ccc(-c3cn(C(C)(C)C)c4ncnc(N)c34)cc2)c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 17/20 0.83
TEK Q02763 17/20 0.83
KDR P35968 13/20 0.83
SRC P12931 12/20 0.80
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
RGS12 O14924 1/20 0.50
NPC1 O15118 1/20 0.50
GMNN O75496 1/20 0.50
ALDH1A1 P00352 1/20 0.50
EGFR P00533 1/20 0.50
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50
FYN P06241 1/20 0.50
LYN P07948 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
MAPT P10636 1/20 0.50
CYP2C9 P11712 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7008467 0.91 LCK (1.00) LCKTEKKDRSRCKDM4E
SCHEMBL7008419 0.90 LCK (0.83) LCKTEKKDRSRCKDM4E
SCHEMBL7011559 0.90 LCK (0.84) LCKTEKKDRSRCKDM4E
SCHEMBL6861193 0.89 LCK (1.00) LCKTEKKDRSRCKDM4E
SCHEMBL7006502 0.89 LCK (0.81) LCKTEKKDRSRCKDM4E
SCHEMBL7009552 0.88 LCK (0.65) LCKTEKKDRSRCEGFR
SCHEMBL7007653 0.86 LCK (0.63) LCKTEKKDRSRCEGFR
SCHEMBL7097902 0.86 KDR (0.63) LCKTEKKDRSRCEGFR
SCHEMBL7008891 0.86 LCK (0.62) LCKTEKKDRSRCEGFR
SCHEMBL7005163 0.86 SRC (0.81) LCKTEKKDRSRCKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970084-B1 PYRROLO 2,3D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS BASF AG (DE) 2003-06-04 EP disclosed
US-6001839-A Substituted 4-amino-7H-pyrrolo [2,3,-d]-pyrimidines as PTK inhibitors BASF AKTIENGESELLSCHAFT (DE) 1999-12-14 US disclosed