SCHEMBL7007305

SCHEMBL7007305

CNc1c(F)cc2c(=O)c(C(=O)O)cn(-c3nc(N)c(F)cc3F)c2c1Cl

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.66
CYP3A4 P08684 2/20 0.66
PIM1 P11309 4/20 0.44
TOP1 P11387 4/20 0.38
ALDH1A1 P00352 3/20 0.38
POLB P06746 3/20 0.38
LMNA P02545 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 1/20 0.38
XBP1 P17861 1/20 0.38
NFKB1 P19838 1/20 0.38
HTT P42858 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
HSD17B10 Q99714 1/20 0.38
EPHA2 P29317 1/20 0.37
FLT4 P35916 1/20 0.37
GSK3B P49841 1/20 0.37
RARB P10826 1/20 0.37
TBXAS1 P24557 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005127 0.90 CYP2C9 (0.58) CYP2C9CYP3A4PIM1TOP1ALDH1A1
SCHEMBL7013484 0.89 CYP2C9 (0.57) CYP2C9CYP3A4PIM1TOP1ALDH1A1
SCHEMBL7010927 0.87 CYP3A4 (0.51) CYP2C9CYP3A4PIM1TOP1ALDH1A1
SCHEMBL7005270 0.87 CYP2C9 (0.60) CYP2C9CYP3A4PIM1TOP1ALDH1A1
SCHEMBL4747757 0.87 CYP2C9 (0.69) CYP2C9CYP3A4PIM1TOP1ALDH1A1
SCHEMBL2670076 0.87 CYP2C9 (0.71) CYP2C9CYP3A4PIM1TOP1ALDH1A1
SCHEMBL14421859 0.86 CYP2C9 (0.66) CYP2C9CYP3A4PIM1TOP1ALDH1A1
SCHEMBL7004218 0.86 CYP2C9 (0.58) CYP2C9CYP3A4PIM1TOP1ALDH1A1
SCHEMBL7007569 0.85 CYP3A4 (0.49) CYP2C9CYP3A4PIM1TOP1ALDH1A1
SCHEMBL7007355 0.85 CYP2C9 (0.60) CYP2C9CYP3A4PIM1TOP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0945435-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed