SCHEMBL7010927

SCHEMBL7010927

CNc1c(F)cc2c(=O)c(C(=O)O)cn(-c3nc(N)ccc3F)c2c1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.51
CYP2C9 P11712 2/20 0.51
PIM1 P11309 3/20 0.48
TOP1 P11387 6/20 0.39
ALDH1A1 P00352 3/20 0.37
POLB P06746 3/20 0.37
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
XBP1 P17861 1/20 0.37
NFKB1 P19838 1/20 0.37
HTT P42858 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TOP2A P11388 6/20 0.36
EPHA2 P29317 1/20 0.36
FLT4 P35916 1/20 0.36
GSK3B P49841 1/20 0.36
RARB P10826 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7007305 0.87 CYP2C9 (0.66) CYP3A4CYP2C9PIM1TOP1ALDH1A1
SCHEMBL7005976 0.87 CYP3A4 (0.55) CYP3A4CYP2C9PIM1TOP1ALDH1A1
SCHEMBL7007569 0.85 CYP3A4 (0.49) CYP3A4CYP2C9PIM1TOP1ALDH1A1
SCHEMBL7008844 0.82 PIM1 (0.56) CYP3A4CYP2C9PIM1TOP1ALDH1A1
SCHEMBL7011977 0.82 TOP1 (0.52) CYP3A4CYP2C9PIM1TOP1ALDH1A1
SCHEMBL7008199 0.80 TOP1 (0.48) CYP3A4CYP2C9PIM1TOP1ALDH1A1
SCHEMBL7851045 0.80 CYP3A4 (0.79) CYP3A4CYP2C9TOP1ALDH1A1POLB
SCHEMBL7010755 0.79 PIM1 (0.46) CYP3A4CYP2C9PIM1TOP1ALDH1A1
SCHEMBL7006342 0.79 PIM1 (0.52) CYP3A4CYP2C9PIM1TOP1ALDH1A1
SCHEMBL7008858 0.79 CYP2C9 (0.47) CYP3A4CYP2C9PIM1TOP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0945435-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed