SCHEMBL7007369

SCHEMBL7007369

Nc1c(F)cc(F)c(-n2cc(C(=O)O)c(=O)c3cc(F)c(Cl)nc32)c1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.46
CYP3A4 P08684 2/20 0.46
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
EPHA2 P29317 1/20 0.41
FLT4 P35916 1/20 0.41
GSK3B P49841 1/20 0.41
RARB P10826 1/20 0.41
TBXAS1 P24557 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
HSD17B10 Q99714 3/20 0.40
LMNA P02545 2/20 0.40
POLB P06746 2/20 0.40
XBP1 P17861 1/20 0.40
NFKB1 P19838 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005531 0.86 STAT3 (0.47) CYP2C9CYP3A4KMT2AKDM4EALDH1A1
SCHEMBL19971429 0.85 KEAP1 (0.48) CYP2C9CYP3A4KEAP1NFE2L2EPHA2
SCHEMBL7013131 0.85 EPHA2 (0.48) CYP2C9CYP3A4KEAP1NFE2L2EPHA2
Hydrochloric Acid SCHEMBL28904892 0.84 KEAP1 (0.47) CYP2C9CYP3A4KEAP1NFE2L2EPHA2
SCHEMBL29980308 0.82 EPHA2 (0.45) CYP2C9CYP3A4KEAP1NFE2L2EPHA2
SCHEMBL19971400 0.82 EPHA2 (0.45) CYP2C9CYP3A4KEAP1NFE2L2EPHA2
SCHEMBL7007504 0.82 EPHA2 (0.47) CYP2C9CYP3A4KEAP1NFE2L2EPHA2
SCHEMBL19973668 0.82 EPHA2 (0.43) CYP2C9CYP3A4KEAP1NFE2L2EPHA2
SCHEMBL19971451 0.82 EPHA2 (0.44) CYP2C9CYP3A4KEAP1NFE2L2EPHA2
SCHEMBL7014638 0.81 EPHA2 (0.44) CYP2C9CYP3A4KEAP1NFE2L2EPHA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787720-B1 PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KK (JP) 2003-07-16 EP disclosed
US-5910498-A NOVEL COMPOUNDS HAVING REDUCED CYTOTOXICITY, PHOTOTOXICITY; TREATING BACTERIAL AND VIRAL INFECTIONS WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1999-06-08 US disclosed
EP-0787720-A1 NOVEL PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1997-08-06 EP disclosed