SCHEMBL7007463

SCHEMBL7007463

NC(=O)OCCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCNCC3)c(F)c21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.62
HPGD P15428 9/20 0.57
HSD17B10 Q99714 9/20 0.57
ALDH1A1 P00352 8/20 0.57
PMP22 Q01453 1/20 0.56
LMNA P02545 4/20 0.52
BRD4 O60885 1/20 0.52
TSHR P16473 1/20 0.52
HTT P42858 1/20 0.52
CYP2J2 P51589 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CYP2C9 P11712 2/20 0.50
ATP6V1B2 P21281 1/20 0.50
TBXA2R P21731 1/20 0.50
EDNRA P25101 1/20 0.50
TARBP2 Q15633 1/20 0.50
TOP2A P11388 5/20 0.48
TOP1 P11387 1/20 0.48
TOP2B Q02880 4/20 0.47
ADRA2B P18089 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10594321 0.90 KDM4E (0.66) KDM4EHPGDHSD17B10ALDH1A1PMP22
SCHEMBL6305606 0.87 KDM4E (0.80) KDM4EHPGDHSD17B10ALDH1A1PMP22
Hydrochloric Acid SCHEMBL10739298 0.86 KDM4E (0.79) KDM4EHPGDHSD17B10ALDH1A1PMP22
Hydrochloric Acid SCHEMBL11187466 0.85 KDM4E (0.68) KDM4EHPGDHSD17B10ALDH1A1PMP22
Hydrochloric Acid SCHEMBL11187784 0.85 KDM4E (0.68) KDM4EHPGDHSD17B10ALDH1A1PMP22
SCHEMBL312379 0.84 KDM4E (0.76) KDM4EHPGDHSD17B10ALDH1A1PMP22
Hydrochloric Acid SCHEMBL10743594 0.83 KDM4E (0.77) KDM4EHPGDHSD17B10ALDH1A1PMP22
Water SCHEMBL10765060 0.83 KDM4E (0.75) KDM4EHPGDHSD17B10ALDH1A1PMP22
SCHEMBL7017181 0.83 KDM4E (0.52) KDM4EHPGDHSD17B10ALDH1A1PMP22
SCHEMBL7007104 0.82 KDM4E (0.63) KDM4EHPGDHSD17B10ALDH1A1PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0614664-B2 Quinolonecarboxylic acid derivatives, their preparation and their use as cell adhesion inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-08 EP disclosed
US-5889009-A ADMINISTERING 1,7-DISUBSTITUTED-4-OX-3-(QUINOLINECARBOXYLIC ACID OR NAPHTHYRIDINECARBOXYLIC ACID) TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-03-30 US disclosed
EP-0614664-B1 Quinolonecarboxylic acid derivatives, their preparation and their use as cell adhesion inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-09-16 EP disclosed
US-5703081-A CELL ADHESION INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-30 US disclosed
US-5519024-A CELL ADHESION INHIBITOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-21 US disclosed
EP-0614664-A1 Quinolonecarboxylic acid derivatives, their preparation and their use as cell adhesion inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-09-14 EP disclosed