SCHEMBL7007590

SCHEMBL7007590

CN(CCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C(=O)[C@H](c1ccccc1)N1CCC(N(CCO)CCCO)CC1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.56
UBE2M P61081 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.40
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39
TACR3 P29371 1/20 0.39
CCR2 P41597 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3472665 1.00 TACR1 (0.56) TACR1UBE2MDCUN1D1SCN5ASCN9A
SCHEMBL7009113 0.93 TACR1 (0.57) TACR1UBE2MDCUN1D1SCN5ASCN9A
SCHEMBL7075456 0.93 TACR1 (0.57) TACR1UBE2MDCUN1D1SCN5ASCN9A
SCHEMBL3473136 0.93 TACR1 (0.53) TACR1UBE2MDCUN1D1SCN5ASCN9A
SCHEMBL3473472 0.93 TACR1 (0.53) TACR1UBE2MDCUN1D1SCN5ASCN9A
SCHEMBL6836873 0.91 TACR1 (0.57) TACR1UBE2MDCUN1D1SCN5ASCN9A
SCHEMBL3475829 0.91 TACR1 (0.57) TACR1UBE2MDCUN1D1SCN5ASCN9A
SCHEMBL5457820 0.84 TACR1 (0.70) TACR1SCN5ASCN9ATACR3
SCHEMBL6836750 0.83 TACR1 (0.58) TACR1UBE2MDCUN1D1SCN5ASCN9A
SCHEMBL3475643 0.83 TACR1 (0.58) TACR1UBE2MDCUN1D1SCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1328516-A1 NOVEL NEUROKININ ANTAGONISTS, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID COMPOUNDS Boehringer Ingelheim Pharma KG (DE) 2003-07-23 EP disclosed
WO-2002032865-A1 NOVEL NEUROKININ ANTAGONISTS, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID COMPOUNDS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2002-04-25 WO disclosed