SCHEMBL7008034

SCHEMBL7008034

CCCCOc1ccc(S(C)(=O)=O)cc1C(=N)SC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 1/20 0.49
LMNA P02545 4/20 0.40
TSHR P16473 3/20 0.40
ADRA2A P08913 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
HTR2B P41595 1/20 0.40
STAT6 P42226 1/20 0.40
KCNH2 Q12809 1/20 0.40
WDR5 P61964 3/20 0.39
BLM P54132 1/20 0.39
SLC6A9 P48067 1/20 0.39
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
MAPT P10636 1/20 0.38
ALPG P10696 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL6633678 0.99 S1PR3 (0.48) S1PR3LMNATSHRADRA2ACYP2D6
SCHEMBL4130038 0.81 S1PR3 (0.71) S1PR3LMNATSHRADRA2ACYP2D6
SCHEMBL6630656 0.80 S1PR3 (0.55) S1PR3LMNATSHRADRA2ACYP2D6
SCHEMBL6630391 0.80 S1PR3 (0.52) S1PR3LMNATSHRADRA2ACYP2D6
Iodide SCHEMBL6627950 0.80 S1PR3 (0.47) S1PR3LMNATSHRADRA2ACYP2D6
SCHEMBL6630509 0.79 S1PR3 (0.54) S1PR3LMNATSHRADRA2ACYP2D6
SCHEMBL4125056 0.77 S1PR3 (0.78) S1PR3LMNAADRA2AHTR2BWDR5
SCHEMBL6630953 0.74 S1PR3 (0.65) S1PR3LMNATSHRADRA2ACYP2D6
SCHEMBL6628554 0.72 S1PR3 (0.49) S1PR3LMNATSHRADRA2ACYP2D6
SCHEMBL4421524 0.70 S1PR3 (0.56) S1PR3LMNATSHRADRA2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368352-A1 CYCLIC GUANOSINE 3',5'-MONOPHOSPHATE PHOSPHODIESTERASE INHIBITORS Pfizer Limited (GB) 2003-12-10 EP disclosed
WO-2002074774-A1 CYCLIC GUANOSINE 3',5'-MONOPHOSPHATE PHOSPHODIESTERASE INHIBITORS PFIZER LIMITED (GB) 2002-09-26 WO disclosed