SCHEMBL7008172

SCHEMBL7008172

CNc1c(F)c(N)c2c(=O)c(C(=O)O)cn(-c3nc(N)c(F)cc3F)c2c1Cl

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.52
CYP2C9 P11712 2/20 0.52
GSK3B P49841 13/20 0.43
TOP2A P11388 1/20 0.39
TOP2B Q02880 1/20 0.39
PIM1 P11309 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
STAT3 P40763 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004180 0.88 CYP3A4 (0.57) CYP3A4CYP2C9GSK3BTOP2ATOP2B
SCHEMBL7012892 0.85 CYP3A4 (0.52) CYP3A4CYP2C9GSK3BTOP2ATOP2B
SCHEMBL7007782 0.85 CYP2C9 (0.54) CYP3A4CYP2C9GSK3BTOP2ATOP2B
SCHEMBL7007305 0.85 CYP2C9 (0.66) CYP3A4CYP2C9GSK3BTOP2ATOP2B
SCHEMBL7858473 0.83 CYP3A4 (0.52) CYP3A4CYP2C9GSK3BTOP2ATOP2B
SCHEMBL7009597 0.83 GSK3B (0.44) GSK3BTOP2ATOP2BPIM1ALDH1A1
SCHEMBL7858346 0.83 CYP3A4 (0.61) CYP3A4CYP2C9GSK3BTOP2ATOP2B
SCHEMBL7857527 0.82 CYP3A4 (0.50) CYP3A4CYP2C9GSK3BTOP2ATOP2B
SCHEMBL7005127 0.81 CYP2C9 (0.58) CYP3A4CYP2C9GSK3BTOP2ATOP2B
SCHEMBL7861219 0.80 CYP3A4 (0.75) CYP3A4CYP2C9GSK3BTOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0945435-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed