SCHEMBL7008267

SCHEMBL7008267

CCC(Oc1ccc(-c2cc3ccccn3c2)cc1)C1CCCNC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.44
NPC1 O15118 2/20 0.39
ALDH1A1 P00352 2/20 0.39
POLB P06746 2/20 0.39
MAPT P10636 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SLC6A2 P23975 3/20 0.33
SLC6A4 P31645 3/20 0.33
PDE6D O43924 1/20 0.33
SLC6A3 Q01959 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6634804 0.86 HRH3 (0.47) HRH3ALDH1A1KDM4ESLC6A2SLC6A4
SCHEMBL6636105 0.82 HRH3 (0.47) HRH3ALDH1A1POLBMAPTSMN1; SMN2
SCHEMBL6633646 0.82 HRH3 (0.46) HRH3ALDH1A1POLBMAPTSMN1; SMN2
SCHEMBL6637128 0.82 HRH3 (0.49) HRH3ALDH1A1POLBMAPTSMN1; SMN2
SCHEMBL6635807 0.80 HRH3 (0.49) HRH3NPC1ALDH1A1MAPTRAB9A
SCHEMBL6635934 0.78 HRH3 (0.50) HRH3ALDH1A1POLBKDM4EMEN1
SCHEMBL28770569 0.77 CYP2D6 (0.38) SLC6A2SLC6A4SLC6A3
SCHEMBL4462917 0.74 SLC6A2 (0.35) SLC6A2SLC6A4SLC6A3
SCHEMBL7008263 0.73 HRH3 (0.58) HRH3NPC1ALDH1A1POLBMAPT
SCHEMBL6642823 0.72 HRH3 (0.56) HRH3NPC1ALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268479-A1 PHENYL-SUBSTITUTED INDOLIZINE DERIVATIVES AND THEIR USE AS HISTAMINE H3 LIGANDS Ortho-McNeil Pharmaceutical, Inc. (US) 2003-01-02 EP claimed
WO-2001074814-A1 PHENYL-SUBSTITUTED INDOLIZINE DERIVATIVES AND THEIR USE AS HISTAMINE H3 LIGANDS ORTHO MCNEIL PHARMACEUTICAL, INC. (US) 2001-10-11 WO claimed