SCHEMBL7008753

SCHEMBL7008753

On1ncc2cccnc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
KDM4D Q6B0I6 1/20 0.44
PARP1 P09874 1/20 0.41
FGFR1 P11362 1/20 0.40
FGFR4 P22455 1/20 0.40
MMP2 P08253 2/20 0.38
TSHR P16473 2/20 0.38
GMNN O75496 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
HSP90AA1 P07900 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
MMP9 P14780 1/20 0.38
ALOX15 P16050 1/20 0.38
NFKB1 P19838 1/20 0.38
MMP8 P22894 1/20 0.38
CCR1 P32246 1/20 0.38
THPO P40225 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14262719 0.76 FGFR1 (0.50) KDM4EKDM4DPARP1FGFR1FGFR4
SCHEMBL21089903 0.75 KDM4E (0.59) KDM4EKDM4DPARP1FGFR1FGFR4
SCHEMBL17114770 0.75 KDM4E (0.55) KDM4EKDM4DPARP1FGFR1FGFR4
SCHEMBL14895754 0.75 KDM4E (0.55) KDM4EKDM4DPARP1FGFR1FGFR4
SCHEMBL3375873 0.75 KDM4E (0.55) KDM4EKDM4DPARP1FGFR1FGFR4
SCHEMBL23227964 0.75 KDM4E (0.55) KDM4EKDM4DPARP1FGFR1FGFR4
SCHEMBL256383 0.75 KDM4E (0.55) KDM4EKDM4DPARP1FGFR1FGFR4
SCHEMBL9935772 0.75 KDM4E (0.50) KDM4EKDM4DPARP1FGFR1FGFR4
SCHEMBL3415322 0.73 KDM4E (0.53) KDM4EKDM4DPARP1FGFR1FGFR4
SCHEMBL31037735 0.73 KDM4E (0.53) KDM4EKDM4DPARP1FGFR1FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0662078-B1 REAGENTS FOR PEPTIDE COUPLINGS RES CORP TECHNOLOGIES INC (US) 2003-05-02 EP disclosed
US-RE38073-E1 Biosynthesis; using dehydration agent RESEARCH CORPORATIONS TECHNOLOGIES, INC. 2003-04-08 US disclosed
US-6534627-B1 Using FMOC (9-fluorenylmethyloxycarbonyl) and tert-butyl containing compounds as protecting group; efficiency and storage stability RESEARCH CORPORATION TECNOLOGIES, INC. 2003-03-18 US disclosed
US-RE37686-E1 Azahydroxybenzotriazoles and derivatives thereof for peptide coupling reactions RESEARCH CORPORATION TECHNOLOGIES, INC. 2002-04-30 US disclosed
US-6040422-A REACTING A FLUOROFORMAMIDINIUM SALT WITH AN N-AMINO PROTECTED, OPTIONALLY SIDE CHAIN PROTECTED AMINO ACID; THEN REACTING PRODUCT WITH A CARBOXY PROTECTED AMINO ACID; FOR COMPOUNDS WITH LONG TERM STORAGE STABILITY RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 2000-03-21 US disclosed
US-5750767-A REACTING PROTECTED AMINO ACID WITH FLUOROFORMAMIDINIUM SALT RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1998-05-12 US disclosed
US-5712418-A FLUOROFORMAMIDINIUM SALTS AS FLUORINATION AGENTS TO FORM PEPTIDES RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1998-01-27 US disclosed
US-5698675-A AMIDATION; ESTERIFICATION RESEARCH CORPORATION TECH., INC. (US) 1997-12-16 US disclosed
US-5644029-A TRIAZOLO-PYRIDINE HETEROCYCLIC COMPOUNDS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1997-07-01 US disclosed
US-5580981-A YELLOW INDICATORS FADING TO COLORLESS UPON COMPLETION OF THE ACYLATION STEP IN AMIDE FORMATION; REACTION ACCELERATORS; LOWERS RACEMIZATION RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1996-12-03 US disclosed
WO-1996004297-A9 SYNTHESIS AND USE OF AMINO ACID FLUORIDES AS PEPTIDE COUPLING REAGENTS 1996-05-02 WO disclosed
WO-1996004297-A1 SYNTHESIS AND USE OF AMINO ACID FLUORIDES AS PEPTIDE COUPLING REAGENTS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1996-02-15 WO disclosed