SCHEMBL7008911

SCHEMBL7008911

Cc1c(Br)cc(CC(N)C(=O)N2CCC(C3CCN(C)CC3)CC2)cc1Br

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 6/20 0.43
OPRK1 P41145 2/20 0.42
OPRD1 P41143 3/20 0.40
ATM Q13315 1/20 0.39
DPP4 P27487 4/20 0.39
HDAC8 Q9BY41 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7008909 1.00 SMYD3 (0.43) SMYD3OPRK1OPRD1ATMDPP4
SCHEMBL7008363 0.91 SMYD3 (0.43) SMYD3OPRK1OPRD1DPP4HDAC8
SCHEMBL7012431 0.88 OPRK1 (0.44) SMYD3OPRK1OPRD1DPP4HDAC8
SCHEMBL7012359 0.81 DPP8 (0.47) SMYD3
SCHEMBL7012362 0.81 DPP8 (0.47) SMYD3
SCHEMBL5658459 0.81 CYP3A4 (0.47) SMYD3
SCHEMBL3279461 0.81 OPRK1 (0.47) SMYD3OPRK1OPRD1DPP4HDAC8
SCHEMBL5891540 0.80 HDAC8 (0.60) OPRK1OPRD1DPP4HDAC8
SCHEMBL7013786 0.79 CALCRL (0.42) SMYD3OPRK1OPRD1HDAC8
SCHEMBL30429936 0.79 DPP4 (0.60) SMYD3OPRK1OPRD1DPP4HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163239-B1 MODIFIED AMINO-ACID AMIDES AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM PHARMA (DE) 2003-05-28 EP disclosed
US-6313097-B1 TREATMENT OR PROPHYLAXIS OF MIGRAINE OR CLUSTER HEADACHES, NON-INSULIN-DEPENDENT DIABETES MELLITUS, INFLAMMATION, ALLERGIC RHINITIS, ASTHMA, MORPHINE TOLERANCE, MENOPAUSAL HOT FLASHES, DISEASES CHARACTERIZED BY EXCESSIVE VASODILATATION BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-11-06 US disclosed