SCHEMBL7009505

SCHEMBL7009505

CC(=O)c1cc(C(=O)Nc2ccc3c(c2)C2CCCN2CCC3)ccc1OC(C)C

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.48
LMNA P02545 1/20 0.48
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
RORC P51449 7/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPT P10636 1/20 0.39
ROCK2 O75116 2/20 0.39
F2 P00734 1/20 0.38
PLG P00747 1/20 0.38
PLAU P00749 1/20 0.38
PLAT P00750 1/20 0.38
KLKB1 P03952 1/20 0.38
PRSS1 P07477 1/20 0.38
CTSS P25774 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7015757 0.99 TP53 (0.47) TP53LMNACNR1CNR2RORC
SCHEMBL7010531 0.96 TP53 (0.44) TP53LMNACNR1CNR2RORC
Hydrochloric Acid SCHEMBL7007356 0.95 TP53 (0.43) TP53LMNACNR1CNR2RORC
SCHEMBL7008605 0.89 RORC (0.42) TP53LMNACNR1CNR2RORC
Hydrochloric Acid SCHEMBL7008692 0.89 RORC (0.41) TP53LMNACNR1CNR2RORC
SCHEMBL7009857 0.88 RORC (0.41) TP53LMNACNR1CNR2RORC
SCHEMBL7012754 0.87 RORC (0.44) CNR1CNR2RORCNPC1RAB9A
Hydrochloric Acid SCHEMBL7010712 0.87 RORC (0.41) TP53LMNACNR1CNR2RORC
SCHEMBL7008091 0.86 RORC (0.40) TP53LMNACNR1CNR2RORC
Hydrochloric Acid SCHEMBL7009820 0.86 RORC (0.44) CNR1CNR2RORCNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102769-B1 TRICYCLIC CARBOXAMIDES SMITHKLINE BEECHAM PLC (GB) 2003-04-16 EP claimed
EP-1102769-B1 TRICYCLIC CARBOXAMIDES SMITHKLINE BEECHAM PLC (GB) 2003-04-16 EP disclosed