SCHEMBL7009599

SCHEMBL7009599

CC(N)OC(=O)c1cn(-c2cc(N)c(F)cc2F)c2c(Cl)c(NCCO)c(F)cc2c1=O

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 3/20 0.40
TOP1 P11387 3/20 0.36
TOP2A P11388 2/20 0.36
ADRB2 P07550 1/20 0.36
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 2/20 0.34
STAT3 P40763 1/20 0.32
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7011913 0.87 PIM1 (0.51) PIM1TOP1TOP2ACYP3A4CYP2C9
Monoethanolamine SCHEMBL7009594 0.85 PIM1 (0.50) PIM1TOP1TOP2ACYP3A4CYP2C9
SCHEMBL7006968 0.85 CYP3A4 (0.50) PIM1TOP1TOP2AADRB2CYP3A4
SCHEMBL7012642 0.82 PIM1 (0.50) PIM1TOP1TOP2AADRB2CYP3A4
SCHEMBL7009088 0.81 PIM1 (0.52) PIM1TOP1TOP2ACYP3A4CYP2C9
SCHEMBL7099804 0.80 PIM1 (0.47) PIM1TOP1TOP2AADRB2CYP3A4
SCHEMBL20912644 0.80 ADRB2 (0.42) PIM1TOP1TOP2AADRB2STAT3
SCHEMBL19728783 0.79 PIM1 (0.49) PIM1TOP1TOP2ACYP3A4CYP2C9
SCHEMBL7009334 0.79 PIM1 (0.48) PIM1TOP1TOP2ACYP3A4CYP2C9
SCHEMBL7011538 0.78 PIM1 (0.51) PIM1TOP1TOP2ACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0945435-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed