SCHEMBL7010093

SCHEMBL7010093

COc1ccc2[nH]cc(C3=CCNCC3)c2n1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.73
ALDH1A1 P00352 4/20 0.73
HSD17B10 Q99714 4/20 0.73
MAPT P10636 3/20 0.73
MEN1 O00255 3/20 0.73
KMT2A Q03164 3/20 0.73
CYP1A2 P05177 2/20 0.73
CYP3A4 P08684 2/20 0.73
CYP2C9 P11712 2/20 0.73
HPGD P15428 2/20 0.73
CYP2C19 P33261 2/20 0.73
HTR2C P28335 4/20 0.57
HTR6 P50406 4/20 0.57
HTR1D P28221 3/20 0.57
MAPK1 P28482 1/20 0.57
BRCA1 P38398 1/20 0.57
DRD2 P14416 1/20 0.49
ALOX15 P16050 1/20 0.49
CYP2D6 P10635 1/20 0.48
HTR1B P28222 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9697117 0.86 KDM4E (0.69) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL9695038 0.86 KDM4E (0.69) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL9695050 0.86 KDM4E (0.83) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL29387209 0.84 KDM4E (1.00) KDM4EALDH1A1HSD17B10MAPTMEN1
Hydrochloric Acid SCHEMBL2159345 0.84 KDM4E (1.00) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL9695044 0.84 KDM4E (1.00) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL9696157 0.83 KDM4E (0.89) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL9696128 0.83 KDM4E (0.64) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL9696693 0.83 KDM4E (0.63) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL9696487 0.80 KDM4E (0.70) KDM4EALDH1A1HSD17B10MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5169947-A 3-(1,2,5,6-tetrahydropyridyl)-pyrrolopyridines PFIZER INC. (US) 1992-12-08 US claimed
EP-0916670-B1 Pyrrolo-(3,2-b) pyridines and their use as 5-HT1F agonists LILLY CO ELI (US) 2003-05-14 EP disclosed
EP-0916670-A2 Pyrrolo-(3,2-b) pyridines and their use as 5-HT1F agonists ELI LILLY AND COMPANY (US) 1999-05-19 EP disclosed
US-5905084-A 5-SUBSTITUTED-3-(PIPERIDIN-4-YL)- AND -3-(1,2,3,6-TETRAHYDROPYRIDIN-4-YL)PYRROLO(3,2-B)PYRIDINES; SIDE EFFECT REDUCTION; NERVOUS SYTEM AND PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY (US) 1999-05-18 US disclosed