SCHEMBL7011985

SCHEMBL7011985

O=C(O)Oc1cn(Cc2nccs2)c2cc(N3CCC(C4CCNCC4)CC3)ccc2c1=O

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 4/20 0.37
KHK P50053 10/20 0.33
KMT2A Q03164 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
CYP3A4 P08684 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
LRRK2 Q5S007 1/20 0.31
ALOX15 P16050 1/20 0.31
ABL1 P00519 1/20 0.31
BCR P11274 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7007290 0.90 TOP1 (0.47) TOP1CNR1CNR2
SCHEMBL7009855 0.85 KHK (0.38) TOP1KHKCNR1CNR2CYP3A4
SCHEMBL7006582 0.81 KDM4E (0.41) TOP1ALOX15
SCHEMBL7011265 0.80 ITGB3 (0.39) KHKCYP3A4ALOX15
SCHEMBL27439565 0.79 FEN1 (0.35) TOP1KHKCYP3A4SMN1; SMN2ALOX15
SCHEMBL7007053 0.74 TOP1 (0.45) TOP1KHKCNR1CNR2
SCHEMBL10804487 0.72 KDM4E (0.50) KHK
Hydrochloric Acid SCHEMBL27411367 0.71 KDM4E (0.36) KHKCYP3A4SMN1; SMN2ALOX15
SCHEMBL7008626 0.70 CHRM1 (0.56) TOP1CNR1CNR2SMN1; SMN2
SCHEMBL7006080 0.70 ITGB3 (0.39) KHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0614664-B2 Quinolonecarboxylic acid derivatives, their preparation and their use as cell adhesion inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-08 EP claimed
EP-0614664-B1 Quinolonecarboxylic acid derivatives, their preparation and their use as cell adhesion inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-09-16 EP claimed