SCHEMBL7012379

SCHEMBL7012379

[CH2]CN1CCCC(Cc2ccc3c(n2)NCCC3)C1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.45
ITGB3 P05106 13/20 0.45
ITGB5 P18084 11/20 0.45
ITGB1 P05556 6/20 0.42
ITGB6 P18564 12/20 0.42
ITGB8 P26012 5/20 0.42
KCNH2 Q12809 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7017295 0.87 ITGAV (0.43) ITGAVITGB3ITGB5ITGB1ITGB6
SCHEMBL7012378 0.81 ITGAV (0.49) ITGAVITGB3ITGB5ITGB1ITGB6
SCHEMBL7397461 0.78 ITGAV (0.47) ITGAVITGB3ITGB5ITGB1ITGB6
SCHEMBL22893988 0.78 ITGAV (0.46) ITGAVITGB3ITGB5ITGB1ITGB6
SCHEMBL30335954 0.76 ITGAV (0.47) ITGAVITGB3ITGB5ITGB1ITGB6
SCHEMBL7007445 0.76 ITGAV (0.47) ITGAVITGB3ITGB5ITGB1ITGB6
SCHEMBL7005713 0.76 ITGAV (0.41) ITGAVITGB3ITGB5ITGB1ITGB6
Hydrochloric Acid SCHEMBL20481212 0.75 ITGAV (0.47) ITGAVITGB3ITGB5ITGB1ITGB6
SCHEMBL7403607 0.75 ITGAV (0.54) ITGAVITGB3ITGB5ITGB1ITGB6
SCHEMBL20139919 0.75 ITGAV (0.46) ITGAVITGB3ITGB5ITGB1ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946165-B1 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2003-04-09 EP disclosed
EP-0946165-A4 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2001-04-11 EP disclosed
EP-0946165-A1 INTEGRIN ANTAGONISTS Merck & Co., Inc. (US) 1999-10-06 EP disclosed
WO-1998018460-A1 INTEGRIN ANTAGONISTS MERCK & CO., INC. (US) 1998-05-07 WO disclosed