SCHEMBL7012940

SCHEMBL7012940

Cc1cccc2nc(C=Cc3ccc(C(=O)c4ccc(C(F)(F)F)cc4)cc3)n(C)c(=O)c12

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
RXFP1 Q9HBX9 1/20 0.43
MAPT P10636 2/20 0.39
TP53 P04637 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39
ADORA2A P29274 2/20 0.38
CYP1A2 P05177 1/20 0.37
MAOB P27338 1/20 0.37
THRB P10828 1/20 0.37
ELANE P08246 1/20 0.37
GFER P55789 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012937 1.00 NPC1 (0.44) NPC1RAB9ARXFP1MAPTTP53
SCHEMBL7014766 0.87 NPC1 (0.58) NPC1RAB9ARXFP1MAPTTP53
SCHEMBL7014764 0.87 NPC1 (0.58) NPC1RAB9ARXFP1MAPTTP53
SCHEMBL7011887 0.84 NPC1 (0.44) NPC1RAB9ARXFP1MAPTTP53
SCHEMBL7011884 0.84 NPC1 (0.44) NPC1RAB9ARXFP1MAPTTP53
SCHEMBL7012661 0.82 NPC1 (0.46) NPC1RAB9ARXFP1MAPTTP53
SCHEMBL7012659 0.82 NPC1 (0.46) NPC1RAB9ARXFP1MAPTTP53
SCHEMBL7015330 0.78 NTRK1 (0.46) NPC1RAB9ASMN1; SMN2MAOBELANE
SCHEMBL7016008 0.77 MEN1 (0.47) RXFP1TP53SMN1; SMN2MAOBALDH1A1
SCHEMBL7017331 0.76 NPC1 (0.44) NPC1RAB9ARXFP1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed