SCHEMBL7014764

SCHEMBL7014764

Cc1cccc2nc(/C=C/c3ccc(C(=O)c4ccc(Cl)cc4)cc3)n(C)c(=O)c12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
RXFP1 Q9HBX9 1/20 0.58
ADORA2A P29274 2/20 0.45
MAOB P27338 1/20 0.45
DRD2 P14416 1/20 0.43
TP53 P04637 2/20 0.42
MAPT P10636 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
DHODH Q02127 1/20 0.41
HTT P42858 2/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7014766 1.00 NPC1 (0.58) NPC1RAB9ARXFP1ADORA2AMAOB
SCHEMBL7012659 0.89 NPC1 (0.46) NPC1RAB9ARXFP1ADORA2AMAOB
SCHEMBL7012661 0.89 NPC1 (0.46) NPC1RAB9ARXFP1ADORA2AMAOB
SCHEMBL7012937 0.87 NPC1 (0.44) NPC1RAB9ARXFP1ADORA2AMAOB
SCHEMBL7011884 0.87 NPC1 (0.44) NPC1RAB9ARXFP1TP53MAPT
SCHEMBL7011887 0.87 NPC1 (0.44) NPC1RAB9ARXFP1TP53MAPT
SCHEMBL7017331 0.78 NPC1 (0.44) NPC1RAB9ARXFP1TP53MAPT
SCHEMBL7012252 0.78 NPC1 (0.37) NPC1RAB9ARXFP1TP53MAPT
SCHEMBL7017333 0.78 NPC1 (0.44) NPC1RAB9ARXFP1TP53MAPT
SCHEMBL7012253 0.78 NPC1 (0.37) NPC1RAB9ARXFP1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed