SCHEMBL7013156

SCHEMBL7013156

COc1ccc(C(=O)c2ccc(CSc3nc4cccc(C)c4c(=O)n3C)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
PTGDR2 Q9Y5Y4 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
LMNA P02545 2/20 0.46
THRB P10828 2/20 0.45
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7011506 0.93 MEN1 (0.55) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7010770 0.91 MEN1 (0.47) DAOHDAC3HDAC4HDAC1HDAC7
SCHEMBL7013547 0.90 PTGDR2 (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7101327 0.90 MEN1 (0.60) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7017586 0.90 MEN1 (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7017967 0.89 DAO (0.52) DAOHDAC3HDAC4HDAC1HDAC7
SCHEMBL7014429 0.89 MEN1 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7015787 0.89 MEN1 (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7013486 0.89 MEN1 (0.45) DAOHDAC3HDAC4HDAC1HDAC7
SCHEMBL7008893 0.89 MEN1 (0.45) DAOHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed