SCHEMBL7013547

SCHEMBL7013547

COC(=O)c1ccc(C(=O)c2ccc(CSc3nc4cccc(C)c4c(=O)n3C)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
DRD2 P14416 1/20 0.50
TBXA2R P21731 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
TSHR P16473 3/20 0.46
MAPK1 P28482 2/20 0.46
MAPT P10636 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
TP53 P04637 3/20 0.46
THRB P10828 1/20 0.45
USP2 O75604 1/20 0.45
NPY1R P25929 1/20 0.45
NPY2R P49146 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7011506 0.93 MEN1 (0.55) PTGDR2MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL7013156 0.90 DAO (0.50) PTGDR2MEN1KMT2ANPC1RAB9A
SCHEMBL7101327 0.90 MEN1 (0.60) PTGDR2MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL7017586 0.90 MEN1 (0.57) PTGDR2MEN1KMT2ASMN1; SMN2TP53
SCHEMBL7015787 0.89 MEN1 (0.51) MEN1KMT2ASMN1; SMN2NPC1MAPT
SCHEMBL7014429 0.89 MEN1 (0.54) MEN1KMT2ADRD2TBXA2RSMN1; SMN2
SCHEMBL7018370 0.88 MEN1 (0.50) PTGDR2MEN1KMT2ADRD2TBXA2R
SCHEMBL7015657 0.88 TP53 (0.52) MEN1KMT2ASMN1; SMN2RAB9AMAPT
SCHEMBL7013147 0.88 MEN1 (0.50) PTGDR2MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL7010770 0.87 MEN1 (0.47) PTGDR2MEN1KMT2ADRD2TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed